Small molecules & peptides
(S)-(+)-GR89696 fumarate
Reference standard for (S)-(+)-[¹¹C]GR89696 (less active enantiomer of the selective κ opioid receptor agonist GR89696)
(S)-(+)-GR89696 fumarate salt; (S)-4-[(3,4-dichlorphenyl)acetyl]-3-(1-pyrrolidinylmethyl)-1-piperazinecarboxylic acid methyl ester fumarate
1-Piperazinecarboxylic acid, 4-[(3,4-dichlorphenyl)acetyl]-3-(1-pyrrolidinylmethyl)-, methyl ester, (S)-, (E)-2-butenedioate (1:1)
Quality
Research Chemical
Characteristics
Molar mass 530.40
CAS RN [150133-21-4]
Purity ≥ 95 %
- Off-white solid
Certificates
CoA: appearance, ¹H and ¹³C NMR spectra
Literature
Ravert H.T. et al. [¹¹C]-GR 89696, a potent kappa opiate receptor radioligand, in vivo binding of the R and S enantiomers. Nuc. Med. Biol. 2002, 29, 47–53.
Talbot P.S. et al. ¹¹C-GR 103545, a Radiotracer for Imaging κ-Opioid Receptors In Vivo with PET: Synthesis and Evaluation in Baboons. J. Nucl. Med. 2005, 46, 484–494.
Naylor A. et al. A Potent New class of κ-Receptor Agonist: 4-Substituted 1-(Arylacetyl)-2-[(dialkylamino)methyl]piperazines. J. Med. Chem. 1993, 36, 2075–2083.
Schoultz B.W. et al. A New Method for Radiosynthesis of ¹¹C-Labeled Carbamate Groups and its Application for a Highly Efficient Synthesis of the Kappa-Opioid Receptor Tracer [¹¹C]GR 103545. The Open Med. Chem. J. 2008, 2 ,72–74.
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| Product | Product No. | Filling amount | Quantity | ||
|---|---|---|---|---|---|
| /products/small-molecules-and-peptides/chemical/598e33db-8c50-4fe5-aaf2-b2363d20412b | Reference Standard | Product No.: 2072 | Filling amount: 1 mg | ||
| /products/small-molecules-and-peptides/chemical/598e33db-8c50-4fe5-aaf2-b2363d20412b | Reference Standard | Product No.: 2072 | Filling amount: 5 mg | ||
| /products/small-molecules-and-peptides/chemical/598e33db-8c50-4fe5-aaf2-b2363d20412b | Reference Standard | Product No.: 2072 | Filling amount: 10 mg | ||
| /products/small-molecules-and-peptides/chemical/598e33db-8c50-4fe5-aaf2-b2363d20412b | Reference Standard | Product No.: 2072 |
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