3-O-Trityl-6-O-desmethyl-buprenorphine
Precursor for 6-O-[¹¹C]-buprenorphine
TDBPN
CA index name: 6,14-Ethenomorphinan-7-methanol, 17-(cyclporopyl-methyl)-α-(1,1-dimethylethyl)-4,5-epoxy-18,19-dihydro-6-hydroxy-α-methyl-3-(triphenylmethoxy)-, (5α, 7α(S))
Quality
Research Chemical
Characteristics
Molar mass 695.93
CAS RN [157891-93-5]
Purity ≥ 95 %
- Colorless to yellowish solid
Certificates
CoA: appearance, ¹H and ¹³C NMR spectra
Literature
Luthra S.K. et al. Automated radiosyntheses of [6-O-methyl-¹¹C]-diprenorphine and [6-O-methyl-¹¹C]buprenorphine from 3-O-trityl protected precursors. Appl. Radiat. Isot. 1994, 45, 857–873.
Luthra S.K. et al. Preparation of [¹¹C]buprenorphine - A potential radioligand for the study of the opiate receptor system in vivo. Int. J. Rad. Appl. Instrum. A. 1987, 38, 65–6.
Lever J.R. et al. Facile synthesis of [¹¹C]buprenorphine for positron emission tomographic studies of opioid receptors. J. Rad. Appl. Instrum. A, 1990, 41, 745–52.
Shiue C.Y. et al. A comparison of the brain uptake of N-(cyclopropyl[¹¹C]methyl)norbuprenorphine ([¹¹C]buprenorphine) and N-(cyclopropyl[¹¹C]methyl)nordiprenorphine ([¹¹C]diprenorphine) in baboon using PET. Int. J. Rad. Appl. Instrum. B, 1991, 18, 281–288.
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Product | Product No. | Filling amount | Quantity | ||
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/products/small-molecules-and-peptides/chemical/8d220f2a-4ea3-4a9d-b1a5-6d8c067e38ad | Precursor | Product No.: 2055 | Filling amount: 1 mg | ||
/products/small-molecules-and-peptides/chemical/8d220f2a-4ea3-4a9d-b1a5-6d8c067e38ad | Precursor | Product No.: 2055 |