Norbinaltorphimine dihydrochloride
NorBNI; N-Desmethylbinaltorphimine; N-Demethylbinaltorphimine dihydrochloride
CA index name: 4,8:11,15-Dimethano-20H-bisbenzofuro[2,3-a:3',2'-i]dipyrido[4,3-b:3',4'-h]carbazole-1,8a,10a,18-tetrol, 7,12-bis(cyclopropylmethyl)-5,6,7,8,9,10,11,12,13,14,19a,20b-dodecahydro-, hydrochloride (1:2), (4bS,8R,8aS,10aS,11R,14aS,19aR,20bR)-
Quality
Research Chemical
Characteristics
Molar mass 734.71
CAS RN [113158-34-2]
Purity ≥ 95 %
- Tan solid
Certificates
CoA: appearance, ¹H NMR spectrum
Literature
Portoghese P.S. et al. Binaltorphimine and nor-binaltorphimine, potent and selective kappa-opioid receptor antagonists. Life Sci. 1987, 40, 1287–1292.
Takemori A.E. et al. Nor-binaltorphimine, a highly selective kappa-opioid antagonist in analgesic and receptor binding assays. J. Pharmacol. Exp. Ther. 1988, 246, 255–258.
Lambert P.D. et al. The effect of central blockade of κ-opioid receptors on neuropeptide Y-induced feeding in the rat. Brain Res. 1993, 629, 146–148.
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Product | Product No. | Filling amount | Quantity | ||
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/products/small-molecules-and-peptides/chemical/d92ffb82-144f-4f3f-99f9-c3e62bc242b3 | Chemicals | Product No.: 4500 | Filling amount: 10 mg | ||
/products/small-molecules-and-peptides/chemical/d92ffb82-144f-4f3f-99f9-c3e62bc242b3 | Chemicals | Product No.: 4500 |