Normethylcarbamoyl-GR 89696
Precursor for [¹¹C]-GR 89696
2-(3,4-Dichlorophenyl)-1-(2-pyrrolidin-1-ylmethyl-piperazine-1-yl)-ethanon; 1-[(3,4-Dichlorophenyl)acetyl]-2-(1-pyrrolidinymethyl)piperazine; Descarbamate-GR 89696
CA index name: Ethanone, 2-(3,4-dichlorophenyl)-1-[2-(1-pyrrolidinylmethyl)-1-piperazinyl]-
Quality
Research Chemical
Characteristics
Molar mass 356.29
CAS RN [126766-48-1]
Purity ≥ 95 %
- Yellowish oil
Certificates
CoA: appearance, ¹H and ¹³C NMR spectra
Literature
Ravert H.T. et al. [¹¹C]-GR 89696, a potent kappa opiate receptor radioligand, in vivo binding of the R and S enantiomers. Nuc. Med. Biol. 2002, 29, 47–53.
Talbot P.S. et al. ¹¹C-GR 103545, a Radiotracer for Imaging κ-Opioid Receptors In Vivo with PET: Synthesis and Evaluation in Baboons. J. Nucl. Med. 2005, 46, 484–494.
Naylor A. et al. A Potent New class of κ-Receptor Agonist: 4-Substituted 1-(Arylacetyl)-2-[(dialkylamino)methyl]piperazines. J. Med. Chem. 1993, 36, 2075–2083.
Schoultz B.W. et al. A New Method for Radiosynthesis of ¹¹C-Labeled Carbamate Groups and its Application for a Highly Efficient Synthesis of the Kappa-Opioid Receptor Tracer [¹¹C]GR 103545. The Open Med. Chem. J. 2008, 2 ,72–74.
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Product | Product No. | Filling amount | Quantity | ||
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/products/small-molecules-and-peptides/chemical/91454850-c1fd-45b6-a679-28cb30e61003 | Precursor | Product No.: 2062 | Filling amount: 1 mg | ||
/products/small-molecules-and-peptides/chemical/91454850-c1fd-45b6-a679-28cb30e61003 | Precursor | Product No.: 2062 | Filling amount: 3 mg | ||
/products/small-molecules-and-peptides/chemical/91454850-c1fd-45b6-a679-28cb30e61003 | Precursor | Product No.: 2062 | Filling amount: 10 mg | ||
/products/small-molecules-and-peptides/chemical/91454850-c1fd-45b6-a679-28cb30e61003 | Precursor | Product No.: 2062 |