EKAP standard
Reference standard for [¹¹C]EKAP
[¹¹C]EKAP standard
Methyl (R)-4-(2-(3,4-dichlorophenyl)acetyl)-3-((diethylamino)methyl)piperazine-1-carboxylate
Quality
Research Chemical
Characteristics
Molar mass 416.34
CAS RN [not yet assigned]
Purity ≥ 95 %
- Colorless to yellow oil
- soluble in dichloromethane, ethyl acetate, dimethyl sulfoxide
Certificates
CoA: ¹H NMR spectrum (identity), HPLC (purity), chiral HPLC (chiral purity)
Literature
Naganawa M. et al. Kinetic modeling and test-retest reproducibility of ¹¹C-EKAP and ¹¹C-FEKAP, novel agonist radiotracers for PET imaging of the κ-opioid receptor in humans. J. Nucl. Med. 2020, 61, 1636–1643.
Li S. et al. Development and In Vivo Evaluation of a κ-Opioid Receptor Agonist as a PET Radiotracer with Superior Imaging Characteristics. J. Nucl. Med. 2019, 60, 1023–1030.
Matuskey D. et al. Social status and demographic effects of the kappa opioid receptor: a PET imaging study with a novel agonist radiotracer in healthy volunteers. Neuropsychopharmacology 2019, 44, 1714–1719.
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Product | Product No. | Filling amount | Quantity | ||
---|---|---|---|---|---|
/products/small-molecules-and-peptides/chemical/c3379d39-0aaa-474e-8ea1-e0d278013c53 | Reference Standard | Product No.: 2075 |