We get the best out of your lead compound

Optimization of lead compounds

We optimize your lead compound, whether this will be a small molecule or a peptide, as a diagnostic or therapeutic radiopharmaceutical. Therefore, we synthesize libraries to optimize structure-activity-relationships in close collaboration with you. We synthesize new molecules around your lead which can be tested in-vitro to obtain further drug candidates. For the most promising compounds we also synthesize primary precursor compounds, considering already optimized leaving/protecting group combinations for high yielding radiolabeling reactions. Our team of medicinal and organic chemists work in state-of-the-art laboratories with optimal equipment to develop your compounds quickly.