6-O-(2-Fluoroethyl)-6-O-desmethyl-phenethyl-orvinol
Reference standard for [¹⁸F]FE-PEO
FE-PEO
CA index name: 6,14-Ethenomorphinan-7-methanol, -4,5-epoxy-6-(2-fluoroethoxy)-α,17-dimethyl-,α-(2-phenylethyl)-3-(triphenylmethoxy)-, (5α, 7α)
Qualität
Research Chemical
Eigenschaften
Molare Masse 505.62
CAS RN [not yet assigned]
Reinheit ≥ 95 %
- Colorless to yellowish solid
Zertifikate
CoA: appearance, ¹H, ¹³C and ¹⁹F NMR spectra
Literatur
Marton J. et al. Design and synthesis of an ¹⁸F-labeled version of phenethyl-orvinol ([¹⁸F]FE-PEO) for PET-imaging of opioid receptors. Molecules 2012, 17, 11554–11569.
Riss P.J. et al. Syntheis and evaluation of ¹⁸F-FE-PEO in rodents: An ¹⁸F-labeled full agonist for opioid receptor imaging. J. Nucl. Med. 2013, 54, 299–305.
Schoultz, B. W. et al. Synthesis and evaluation of three structurally related ¹⁸F-labeled orvinols of different intrinsic activities: [¹⁸F]fluoroethyl-diprenorphine ([¹⁸F]FDPN), [¹⁸F]fluoroethyl-buprenorphine ([¹⁸F]FBPN and [¹⁸F]fluoroethyl-phenethyl-orvinol ([¹⁸F]FPEO. J. Med. Chem. 2014, 57, 5464–5469.
Zur Anfrage hinzufügen
Produkt | Produktnummer | Füllmenge | Anzahl | ||
---|---|---|---|---|---|
/de/Produkte/Kleine-Molekuele-und-Peptide/chemical/4164c3db-8be8-435a-8863-23f593e8947a | Reference Standard | Produktnummer: 2053 | Füllmenge: 10 mg | ||
/de/Produkte/Kleine-Molekuele-und-Peptide/chemical/4164c3db-8be8-435a-8863-23f593e8947a | Reference Standard | Produktnummer: 2053 |